Cepacol Maximum Strength Menthol

Cepacol Maximum Strength Menthol Uses, Dosage, Side Effects, Food Interaction and all others data.

Cepacol Maximum Strength Menthol, an ester local anaesthetic, blocks the initiation and conduction of nerve impulses by decreasing the neuronal membrane’s permeability to Na ions, which results in inhibition of depolarisation with resultant blockade of conduction.

Cepacol Maximum Strength Menthol is indicated for use as a topical anesthetic. It has a duration of action of approximately 10 minutes and a wide therapeutic window. Patients should be counselled regarding the risks of methemoglobinemia.

Trade Name Cepacol Maximum Strength Menthol
Generic Benzocaine
Benzocaine Other Names Amben ethyl ester, Benzocaina, Benzocaine, Benzocainum, Ethyl aminobenzoate, Ethyl p-aminobenzoate, Ethyl p-aminophenylcarboxylate, p-(Ethoxycarbonyl)aniline, p-Carbethoxyaniline, p-Ethoxycarboxylic aniline
Type Mucous membrane gel, mucous membrane liquid, mucous membrane paste, mucous membrane powder for reconstitution, mucous membrane spray, mucous membrane swab, mucous membrane tablet, disintegrating, rectal ointment, topical cream, topical gel, topical liquid, topical lotion, topical ointment, topical spray, topical stick, topical swab
Formula C9H11NO2
Weight Average: 165.1891
Monoisotopic: 165.078978601
Protein binding

Benzocaine binds to both serum albumin and alpha-1-acid glycoprotein.

Groups Approved, Investigational
Therapeutic Class Local & Surface anesthesia
Manufacturer
Available Country United States
Last Updated: September 19, 2023 at 7:00 am
Cepacol Maximum Strength Menthol
Cepacol Maximum Strength Menthol

Uses

For the temporary relief of pain due to minor injury or irritation of the mouth and gums like Toothache, Sore gums, Canker sores, Braces, Minor dental procedures, Dentures

Cepacol Maximum Strength Menthol is also used to associated treatment for these conditions: Acute Sore Throat Pain, Dental Pain, Gangrene Stomatitis, Gingivitis, Hemorrhoids, Laryngitis, Pharyngitis, Premature Ejaculation, Secondary Bacterial Infection caused by Tonsillectomy, Secondary Bacterial Infection caused by Tooth Extractions, Skin Irritation, Sore Throat, Stomatitis, Sunburn, Teething pain, Tonsillitis, Tooth Pain, Vomiting, Pruritic dermatosis, Ulceration of the mouth, Buccopharyngeal anesthesia

How Cepacol Maximum Strength Menthol works

Cepacol Maximum Strength Menthol diffuses into nerve cells where it binds to sodium channels, preventing the channels from opening, and blocking the influx of sodium ions. Nerve cells unable to allow sodium into cells cannot depolarize and conduct nerve impulses.

Dosage

Cepacol Maximum Strength Menthol dosage

Apply to the affected area up to 4 times daily or as directed by a doctor/dentist. Children under 12 years of age should be supervised during the use of this product. Children under 2 years of age should be consulted to a doctor/dentist prior to the use of this product. An easy application might be done by fixing applicator on the tube’s nozzle. After application, supplied cap should be fixed on top of the applicator.

Side Effects

Side effects are less common. The side effects include allergies, swelling in the mouth or throatetc.

Toxicity

Patients experiencing an overdose may present with local anesthetic systemic toxicity syndrome, decreased cardiovascular function, decreased central nervous system function, cardiac arrest, bradycardia, hypotension, cardiac arrhythmias, syncope, and seizures. Patients should be treated with symptomatic and supportive measures which include airway maintenance, controlling seizures, and hemodynamic stabilization.

Precaution

Patient with asthma, bronchitis, emphysema, heart disease; smokers. Children, Pregnancy and lactation.

Interaction

May antagonise the therapeutic effect of sulfonamides. Anticholinesterases may inhibit the metabolism benzocaine.

Food Interaction

No interactions found.

Pregnancy & Breastfeeding use

Pregnancy Category C. Either studies in animals have revealed adverse effects on the fetus (teratogenic or embryocidal or other) and there are no controlled studies in women or studies in women and animals are not available. Drugs should be given only if the potential benefit justifies the potential risk to the fetus.

Contraindication

Epiglottis (oral spray), methaemoglobinaemia.

Acute Overdose

Symptom: Methaemoglobinaemia, manifested by cyanotic (greyish) skin discolouration, unusual breathing or breathlessness.

Management: Symptomatic and supportive treatment. IV methylene blue 1% may be administered.

Storage Condition

Store between 15-30° C.

FAQ

What is Cepacol Maximum Strength Menthol used for?

Cepacol Maximum Strength Menthol topical is used to reduce pain or discomfort caused by minor skin irritations, sore throat, sunburn, vaginal or rectal irritation, ingrown toenails, hemorrhoids, and many other sources of minor pain on a surface of the body. Cepacol Maximum Strength Menthol is an ester local anesthetic commonly used as a topical pain reliever or in cough drops. It is the active ingredient in many over-the-counter anesthetic ointments such as products for oral ulcers.

How safe is Cepacol Maximum Strength Menthol?

Cepacol Maximum Strength Menthol topical used in the mouth may cause a condition in which the oxygen in your body tissues can become dangerously low. This is a potentially fatal condition called methemoglobinemia. Do not use Cepacol Maximum Strength Menthol topical if you have ever had methemoglobinemia.

How does Cepacol Maximum Strength Menthol work?

Cepacol Maximum Strength Menthol works by blocking nerve signals in your body.

What are the common side effects of Cepacol Maximum Strength Menthol?

Common side effects of Cepacol Maximum Strength Menthol are include:

  • Bluish-colored lips, fingernails, or palms.
  • difficulty breathing.
  • dizziness or lightheadedness.
  • high fever.
  • rapid heart rate.
  • worsening of pain, redness, swelling, or irritation in or around the mouth.

Is Cepacol Maximum Strength Menthol safe during pregnancy?

Cepacol Maximum Strength Menthol topical is only recommended for use during pregnancy when benefit outweighs risk.

Is Cepacol Maximum Strength Menthol safe during breastfeeding?

Cepacol Maximum Strength Menthol has not been studied during breastfeeding, but is unlikely to affect her breastfed infant if it is applied away from the breast.

Can I drink alcohol with Cepacol Maximum Strength Menthol?

Alcohol and Cepacol Maximum Strength Menthol creates a that has different effects depending on the dose: many people feel stimulated and strengthened at low doses of alcohol and Cepacol Maximum Strength Menthol and even mixing a small amount of Cepacol Maximum Strength Menthol and alcohol is not recommended.

How often can I take Cepacol Maximum Strength Menthol?

Do not use the Cepacol Maximum Strength Menthol more than four times a day.

How should I use Cepacol Maximum Strength Menthol topical?

Use exactly as directed on the label, or as prescribed by your doctor. Read all medication guides or instruction sheets. Your body may absorb more of benzocaine topical if you use too much, if you apply it over large skin areas, or if you apply heat, bandages, or plastic wrap to treated skin areas. Skin that is cut or irritated may also absorb more topical medication than healthy skin.

How long does Cepacol Maximum Strength Menthol take to work?

Cepacol Maximum Strength Menthol is a water-insoluble ester-type local anesthetic agent that is mainly useful for topical application. The onset of action is rapid (<1 minute), and the effective duration is 5 to 10 minutes. 

What happens if I use Cepacol Maximum Strength Menthol too much?

An overdose of Cepacol Maximum Strength Menthol topical applied to the skin can cause life-threatening side effects such as uneven heartbeats, seizure (convulsions), coma, slowed breathing, or respiratory failure (breathing stops).

How much Cepacol Maximum Strength Menthol is toxic?

The threshold toxic dose for Cepacol Maximum Strength Menthol is 22-40 mg/kg.

Who should not take Cepacol Maximum Strength Menthol?

Do not use benzocaine topical if you have ever had methemoglobinemia. Do not use Cepacol Maximum Strength Menthol topical on a child younger than 2 years old.

What happens if I miss a dose?

Since Cepacol Maximum Strength Menthol topical is used when needed, you may not be on a dosing schedule. Skip any missed dose if it's almost time for your next dose.

What what happen if I overdose?

Seek emergency medical attention. An overdose of benzocaine topical applied to the skin can cause life-threatening side effects such as uneven heartbeats, seizure (convulsions), coma, slowed breathing, or respiratory failure (breathing stops).

Will Cepacol Maximum Strength Menthol affect my fertility?

Studies have not been done to see if Cepacol Maximum Strength Menthol could affect male fertility or increase the chance of birth defects. In general, exposures that fathers or sperm donors have are unlikely to increase the risks to a pregnancy.

Can I drive after taking Cepacol Maximum Strength Menthol ?

Cepacol Maximum Strength Menthol does not affect your ability to drive.

Can Cepacol Maximum Strength Menthol affects my liver?

Please consult your doctor if you have any concerns regarding the usage of Cepacol Maximum Strength Menthol in patients with liver impairment.

Can Cepacol Maximum Strength Menthol affects my kidney?

Please consult your doctor if you have any concerns regarding the usage of Cepacol Maximum Strength Menthol in patients with kidney impairment.

Can I take Cepacol Maximum Strength Menthol for a long time?

Cepacol Maximum Strength Menthol should not be used for longer durations unless prescribed by a doctor. If your condition does not improve despite using Cepacol Maximum Strength Menthol for a week, consult your doctor, he/she may prescribe you an alternate medicine.

Is It safe to use Cepacol Maximum Strength Menthol on large areas of skin?

The topical form of Cepacol Maximum Strength Menthol should not be used on large areas of skin, deep puncture wounds, raw or blistered skin, and on severe burns or abrasions. Use the smallest amount of Cepacol Maximum Strength Menthol to numb the skin and to relieve pain.

Is Cepacol Maximum Strength Menthol safe to treat mouth ulcers ?

Cepacol Maximum Strength Menthol  is used to treat mouth ulcers, canker sores and mouth irritation. Mouth ulcers, also known as canker sores are small, painful lesions which develop in the mouth or at the base of gums.

Can Cepacol Maximum Strength Menthol be used for teething pain?

Cepacol Maximum Strength Menthol should not be used to treat teething pain in infants.

can I eat after using Cepacol Maximum Strength Menthol?

If you are using Cepacol Maximum Strength Menthol for treating tooth pain, gum pain, or mouth ulcers, avoid eating within 1hour after using Cepacol Maximum Strength Menthol. Cepacol Maximum Strength Menthol numbs the skin; this might cause biting of the tongue. Avoid swallowing the topical form of Cepacol Maximum Strength Menthol while applying it to your gums or inside the mouth.

*** Taking medicines without doctor's advice can cause long-term problems.
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