Cinolazepamum
Cinolazepamum Uses, Dosage, Side Effects, Food Interaction and all others data.
Cinolazepamum is a benzodiazepine derivative with anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant activity. It is not approved in Canada or America.
Trade Name | Cinolazepamum |
Generic | Cinolazepam |
Cinolazepam Other Names | Cinolazepam, Cinolazepamum |
Type | |
Formula | C18H13ClFN3O2 |
Weight | Average: 357.766 Monoisotopic: 357.068032587 |
Groups | Experimental |
Therapeutic Class | |
Manufacturer | |
Available Country | |
Last Updated: | September 19, 2023 at 7:00 am |
Uses
Cinolazepamum is a benzodiazepine used to manage severe and debilitating forms of sleep disorders of various origins in adults.
For the management of anxiety disorders or for the short-term relief of the symptoms of anxiety or anxiety associated with depressive symptoms.
Cinolazepamum is also used to associated treatment for these conditions: Insomnia, Sleep Disorder
How Cinolazepamum works
Cinolazepamum binds to central benzodiazepine receptors which interact allosterically with GABA receptors. This potentiates the effects of the inhibitory neurotransmitter GABA, increasing the inhibition of the ascending reticular activating system and blocking the cortical and limbic arousal that occurs following stimulation of the reticular pathways.
Toxicity
The onset of impairment of consciousness is relatively rapid in benzodiazepine poisoning. Onset is more rapid following larger doses and with agents of shorter duration of action. The most common and initial symptom is somnolence. This may progress to coma Grade I or Grade II following very large ingestions.
Food Interaction
- Avoid alcohol.
- Limit caffeine intake.
- Take with food.
Elimination Route
Bioavailability following oral administration is 90-100%.
Half Life
9 hours
Innovators Monograph
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