Balarsen Uses, Dosage, Side Effects and more

Balarsen (INN) is an antiprotozoal agent that was first synthesized by Ernst A.H. Friedheim in 1949 via the complexing of acetarsol with 2,3-dimercaptopropanol. It has since been demonstrated that the agent possesses activity against amoebas and yaws. Considered well tolerated when compared to other related trivalent organoarsenicals, arsthinol has even undergone recent studies as a potential anticancer agent.

Trade Name Balarsen
Generic Arsthinol
Arsthinol Other Names Arsthinenol, Arsthinol
Type
Formula C11H14AsNO3S2
Weight Average: 347.285
Monoisotopic: 346.963106116
Groups Experimental
Therapeutic Class
Manufacturer
Available Country
Last Updated: January 7, 2025 at 1:49 am

Uses

Antiprotozoal agent effective against amoebiasis and yaws.

Toxicity

Oral,mouse: LD50 = 300 mg/kg; Oral, rabbit: LD50 = 3200 mg/kg; Oral, rat: LD50 = 980 mg/kg.

Innovators Monograph

*** Taking medicines without doctor's advice can cause long-term problems.
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