Cinalukast

Cinalukast Uses, Dosage, Side Effects, Food Interaction and all others data.

Used in the treatment of asthma, cinalukast selectively antagonizes leukotriene D4 (LTD4) at the cysteinyl leukotriene receptor, CysLT1, in the human airway. Cinalukast inhibits the actions of LTD4 at the CysLT1 receptor, preventing airway edema, smooth muscle contraction, and enhanced secretion of thick, viscous mucus.

Trade Name Cinalukast
Generic Cinalukast
Cinalukast Other Names Cinalukast
Type
Formula C23H28N2O3S
Weight Average: 412.545
Monoisotopic: 412.182063462
Groups Experimental
Therapeutic Class
Manufacturer
Available Country
Last Updated: September 19, 2023 at 7:00 am
Cinalukast
Cinalukast

Uses

For Protection against second- phase inflamation in exercise-induced bronchoconstriction and Asthma.

How Cinalukast works

Binds to the cysteinyl leukotriene receptor. The cysteinyl leukotrienes (LTC4, LTD4, LTE4) are products of arachidonic acid metabolism and are released from various cells, including mast cells and eosinophils. These eicosanoids bind to cysteinyl leukotriene receptors (CysLT) found in the human airway. Cysteinyl leukotrienes and leukotriene receptor occupation have been correlated with the pathophysiology of asthma, including airway edema, smooth muscle contraction, and altered cellular activity associated with the inflammatory process, which contribute to the signs and symptoms of asthma.

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*** Taking medicines without doctor's advice can cause long-term problems.
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