Mirfentanil Uses, Dosage, Side Effects and more

Mirfentanil is a derivative of fentanyl that presents high selectivity for the mu opioid receptor. At lower doses, it antagonizes the analgesic effects of alfentanil and substitutes for naloxone in morphine-treated monkeys; however, it also reverses naloxone-precipitated withdrawal in pigeons trained to discriminate morphine from naloxone. At high doses, it exhibits analgesic activity which is not fully reversed by opioid antagonists, suggesting that the drug has both opioid and non-opioid mechanisms of action.

Trade Name Mirfentanil
Generic Mirfentanil
Mirfentanil Other Names Mirfentanil
Type
Formula C22H24N4O2
Weight Average: 376.46
Monoisotopic: 376.189926029
Groups Experimental
Therapeutic Class
Manufacturer
Available Country
Last Updated: January 7, 2025 at 1:49 am

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