SR 121463
SR 121463 Uses, Dosage, Side Effects, Food Interaction and all others data.
SR 121463 is a nonpeptide aquaretic compound with potent selective antagonism of the vasopressin V2 (V1b) receptor subtype. It is a candidate for control of hyponatremia and in the treatment of syndrome of inappropriate secretion of anti-diuretic hormone (SIADH).
Increases urine volume through selective antagonism of V1b/V2 receptors.
Trade Name | SR 121463 |
Generic | SR 121463 |
Type | |
Groups | Investigational |
Therapeutic Class | |
Manufacturer | |
Available Country | |
Last Updated: | September 19, 2023 at 7:00 am |
Uses
Investigated for use/treatment in cardiovascular disorders, in the treatment of syndrome of inappropriate secretion of anti-diuretic hormone (SIADH) and in hyponatremia.
How SR 121463 works
Selectively antagonizes v1b receptors.
Toxicity
Phase 11b showed a good clinical safety profile.
Innovators Monograph
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