Telapristone acetate Uses, Dosage, Side Effects and more
Telapristone acetate, an orally-available, selective progesterone receptor modulator, is in development to alleviate symptoms associated with both uterine fibroids and endometriosis.
Patients receiving Proellex saw improvements in key symptoms associated with uterine fibroids, namely reduced pain and bleeding, as well as effects on bone retention.
| Trade Name | Telapristone acetate |
| Generic | Telapristone acetate |
| Telapristone acetate Other Names | Telapristone acetate |
| Type | |
| Formula | C31H39NO5 |
| Weight | Average: 505.655 Monoisotopic: 505.28282336 |
| Groups | Investigational |
| Therapeutic Class | |
| Manufacturer | |
| Available Country | |
| Last Updated: | January 7, 2025 at 1:49 am |
Uses
For the treatment of uterine fibroids and endometriosis.
How Telapristone acetate works
Proellex selectively blocks the progesterone receptor thus avoiding the adverse effects of GnRH agonists associated with the induction of a low estrogen, menopausal-like state in women.
Elimination Route
Orally-available
