Bupranolol

Bupranolol Uses, Dosage, Side Effects, Food Interaction and all others data.

Bupranolol is a non-selective beta blocker with potency similar to propanolol. It does not have intrinsic sympathomimetic activity (ISA), but does have strong membrane stabilizing activity.

Bupranolol is a competitive, nonselective beta-blocker similar to propanolol without intrinsic sympathomimetic activity.

Table Of contents

• Bupranolol
• Uses
• Dosage
• Side Effect
• Precautions
• Interactions
• Uses during Pregnancy
• Uses during Breastfeeding
• Accute Overdose
• Food Interaction
• Half Life
• Volume of Distribution
• Clearance
• Interaction With other Medicine
• Contradiction
• Storage

Trade Name	Bupranolol
Generic	Bupranolol
Bupranolol Other Names	Bupranolol, Bupranololum
Type
Formula	C14H22ClNO2
Weight	Average: 271.783 Monoisotopic: 271.13390666
Protein binding	76%
Groups	Experimental
Therapeutic Class
Manufacturer
Available Country
Last Updated:	September 19, 2023 at 7:00 am

Uses

Used to manage hypertension and tachycardia. Also used to treat glaucoma.

How Bupranolol works

Bupranolol competes with sympathomimetic neurotransmitters such as catecholamines for binding at beta(1)-adrenergic receptors in the heart, inhibiting sympathetic stimulation. This results in a reduction in resting heart rate, cardiac output, systolic and diastolic blood pressure, and reflex orthostatic hypotension.

Toxicity

Symptoms of overdose include bradycardia, cardiac failure, hypotension, and brochospasm.

Elimination Route

Quickly and completely absorbed from the gut with less than 10% oral bioavailability.

Half Life

2-4 hours

Innovators Monograph

You find simplified version here Bupranolol