Bupranololum
Bupranololum Uses, Dosage, Side Effects, Food Interaction and all others data.
Bupranololum is a non-selective beta blocker with potency similar to propanolol. It does not have intrinsic sympathomimetic activity (ISA), but does have strong membrane stabilizing activity.
Bupranololum is a competitive, nonselective beta-blocker similar to propanolol without intrinsic sympathomimetic activity.
Trade Name | Bupranololum |
Generic | Bupranolol |
Bupranolol Other Names | Bupranolol, Bupranololum |
Type | |
Formula | C14H22ClNO2 |
Weight | Average: 271.783 Monoisotopic: 271.13390666 |
Protein binding | 76% |
Groups | Experimental |
Therapeutic Class | |
Manufacturer | |
Available Country | |
Last Updated: | September 19, 2023 at 7:00 am |
Uses
Used to manage hypertension and tachycardia. Also used to treat glaucoma.
How Bupranololum works
Bupranololum competes with sympathomimetic neurotransmitters such as catecholamines for binding at beta(1)-adrenergic receptors in the heart, inhibiting sympathetic stimulation. This results in a reduction in resting heart rate, cardiac output, systolic and diastolic blood pressure, and reflex orthostatic hypotension.
Toxicity
Symptoms of overdose include bradycardia, cardiac failure, hypotension, and brochospasm.
Elimination Route
Quickly and completely absorbed from the gut with less than 10% oral bioavailability.
Half Life
2-4 hours
Innovators Monograph
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