MedicinesFAQ

Amuvatinib Uses, Dosage, Side Effects and more

Amuvatinib has been used in trials studying the treatment of Solid Tumors and Small Cell Lung Carcinoma. Amuvatinib is an oral, selective multi-targeted tyrosine kinase inhibitor that suppresses c-MET, c-RET and the mutant forms of c-KIT, PDGFR and FLT3. Amuvatinib also suppresses Rad51 protein, a critical component of double-stranded DNA repair in cancer cells.

Attribute Details
Trade Name Amuvatinib
Generic Amuvatinib
Amuvatinib Other Names Amuvatinib
Type
Formula C23H21N5O3S
Weight Average: 447.51
Monoisotopic: 447.13651073
Groups Investigational
Therapeutic Class
Manufacturer
Available Country
Last Updated: January 7, 2025 at 1:49 am
   

Uses

Amuvatinib is a selective multi-targeted tyrosine kinase inhibitor that suppresses c-MET, c-RET and the mutant forms of c-KIT, PDGFR and FLT3. Amuvatinib also suppresses Rad51 protein, a critical component of double-stranded DNA repair in cancer cells.

Elimination Route

Orally available

Innovators Monograph

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