MedicinesFAQ

Quizartinibum Uses, Dosage, Side Effects and more

Quizartinibum is under investigation in Childhood Acute Myeloid Leukemia/Other Myeloid Malignancies. It is a potent inhibitor of FLT3.

In preclinical studies, Quizartinibum demonstrated dose-dependent activity and favorable drug-like profiles in bioavailability, pharmacokinetics, cytochrome P450 (CYP) liability, and absorption, distribution, metabolism, excretion (ADME).

Attribute Details
Trade Name Quizartinibum
Generic Quizartinib
Quizartinib Other Names Quizartinib, Quizartinibum
Type
Formula C29H32N6O4S
Weight Average: 560.67
Monoisotopic: 560.220574708
Groups Investigational
Therapeutic Class
Manufacturer
Available Country
Last Updated: January 7, 2025 at 1:49 am
   

How Quizartinibum works

Quizartinibum potently inhibits FLT3, a kinase that is mutated in approximately one-third of acute myeloid leukemia cases, and patients with FLT3 mutations are less responsive to traditional therapies.

Innovators Monograph

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